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CP-809101 hydrochloride
CAS No. 1215721-40-6
CP-809101 hydrochloride ( —— )
Catalog No. M26127 CAS No. 1215721-40-6
CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 41 | In Stock |
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| 5MG | 68 | In Stock |
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| 10MG | 105 | In Stock |
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| 25MG | 232 | In Stock |
|
| 50MG | 431 | In Stock |
|
| 100MG | 617 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCP-809101 hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionCP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).
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DescriptionCP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).(In Vitro):CP-809101 is a potent, functionally selective 5-HT2C agonist that displays approximately 100% efficacy in vitro.(In Vivo):Similar to currently available antipsychotic drugs, CP-809101 dose-dependently inhibited conditioned avoidance responding (CAR, ED50 = 4.8 mg/kg, sc). CP-809101 antagonized both PCP- and d-amphetamine-induced hyperactivity with ED50 values of 2.4 and 2.9 mg/kg (sc), respectively, and also reversed an apomorphine induced-deficit in prepulse inhibition. At doses up to 56 mg/kg, CP-809101 did not produce catalepsy. CP-809101 was inactive in two animal models of antidepressant-like activity, the forced swim test, and learned helplessness.
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Synonyms——
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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RecptorNMDA
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Research Area——
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Indication——
Chemical Information
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CAS Number1215721-40-6
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Formula Weight341.2
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Molecular FormulaC15H18Cl2N4O
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Purity>98% (HPLC)
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Solubility——
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SMILESCl.Clc1cccc(COc2cncc(n2)N2CCNCC2)c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Mikolajczak P et al. Effects of acamprosate and some polyamine site ligands of NMDA receptor on short-term memory in rats. Eur J Pharmacol. 2002 May 24;444(1-2):83-96.
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